umbralisib (TGR-1202) - CD BioSciences

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umbralisib (TGR-1202)

umbralisib (TGR-1202)

SPC-02301

umbralisib (TGR-1202)

CAS No. 1532533-67-7

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PI3K inhibitor

Description
TGR-1202, a novel, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 & 24.3 nM, respectively.
Product Details
CAS No. CAS No. 1532533-67-7
Description TGR-1202, a novel, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 & 24.3 nM, respectively.
Formula C31H24F3N5O3
Molecular Weight 571.55
Storage 3 years -20°C powder
2 years -80°C in solvent
Synonyms Rp-5264
SMILES CC(C)OC1=C(C=C(C=C1)C2=NN(C3=NC=NC(=C23)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F
Usage
Storage 3 years -20°C powder
2 years -80°C in solvent

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